Carbonium vs. carbenium ion-like transition state geometries for carbocation cyclization - how strain associated with bridging affects 5-exo vs. 6-endo selectivity.

نویسندگان

  • Osvaldo Gutierrez
  • Jason G Harrison
  • Ryan J Felix
  • Fernando Cortés Guzman
  • Michel R Gagné
  • Dean J Tantillo
چکیده

Quantum chemical calculations are used to explore the origins of regioselectivity for proton-, Pt(II)- and Pd(II)-promoted cyclizations of 1,5-hexadienes, 5-aminoalkenes, and allylic acetimidates. The strain associated with achieving carbonium ion-like transition state geometries is shown to be a key factor in controlling 5-exo vs. 6-endo selectivity.

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عنوان ژورنال:
  • Chemical science

دوره 4 10  شماره 

صفحات  -

تاریخ انتشار 2013